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Tyrphostin AG1433

CAS No. 168835-90-3

Tyrphostin AG1433 ( SU1433; AG1433 )

产品货号. M26493 CAS No. 168835-90-3

Tyrphostin AG1433 is an inhibitor of tyrosine kinases and also a dual inhibitor of PDGFRβ(IC50s = 5.0 μM) and VEGFR-2 (Flk-1/KDR)(IC50s = 9.3 μM).

纯度: >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
规格 价格/人民币 库存 数量
2MG ¥599 有现货
5MG ¥988 有现货
10MG ¥1596 有现货
25MG ¥2859 有现货
50MG ¥4358 有现货
100MG ¥6302 有现货
500MG ¥12879 有现货
1G 获取报价 有现货

生物学信息

  • 产品名称
    Tyrphostin AG1433
  • 注意事项
    本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
  • 产品简述
    Tyrphostin AG1433 is an inhibitor of tyrosine kinases and also a dual inhibitor of PDGFRβ(IC50s = 5.0 μM) and VEGFR-2 (Flk-1/KDR)(IC50s = 9.3 μM).
  • 产品描述
    Tyrphostin AG1433 is an inhibitor of tyrosine kinases and also a dual inhibitor of PDGFRβ(IC50s = 5.0 μM) and VEGFR-2 (Flk-1/KDR)(IC50s = 9.3 μM).(In Vitro):In glioblastoma cells, administration of Tyrphostin AG1433 (0.1-100 μM; 72 hours; GB8B cells) induces moderate cytotoxicity .(In Vivo):Tyrphostin AG1433 is prepared in methylcellulose pellets and applies to the CAMs of 4-6-day-old chicken embryos, and prevents the formation of new vessels under the pellets .
  • 同义词
    SU1433; AG1433
  • 通路
    Angiogenesis
  • 靶点
    VEGFR
  • 受体
    ——
  • 研究领域
    ——
  • 适应症
    ——

化学信息

  • CAS Number
    168835-90-3
  • 分子量
    266.3
  • 分子式
    C16H14N2O2
  • 纯度
    >98% (HPLC)
  • 溶解度
    ——
  • SMILES
    OC1=CC=C(C2=NC3=CC(C)=C(C)C=C3N=C2)C=C1O
  • 化学全称
    ——

运输与储存

  • 储存条件
    (-20℃)
  • 运输条件
    With Ice Pack
  • 稳定性
    ≥ 2 years

参考文献

1.Shuyun Shi, et al. A high-speed counter-current chromatography- HPLC-DAD method for preparative isolation and purification of two polymethoxylated flavones from Taraxacum mongolicum. J Chromatogr Sc . May-Jun 2009;47(5):349-53.
产品手册
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