Tyrphostin AG1433
CAS No. 168835-90-3
Tyrphostin AG1433 ( SU1433; AG1433 )
产品货号. M26493 CAS No. 168835-90-3
Tyrphostin AG1433 is an inhibitor of tyrosine kinases and also a dual inhibitor of PDGFRβ(IC50s = 5.0 μM) and VEGFR-2 (Flk-1/KDR)(IC50s = 9.3 μM).
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
规格 | 价格/人民币 | 库存 | 数量 |
2MG | ¥599 | 有现货 |
|
5MG | ¥988 | 有现货 |
|
10MG | ¥1596 | 有现货 |
|
25MG | ¥2859 | 有现货 |
|
50MG | ¥4358 | 有现货 |
|
100MG | ¥6302 | 有现货 |
|
500MG | ¥12879 | 有现货 |
|
1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称Tyrphostin AG1433
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注意事项本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
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产品简述Tyrphostin AG1433 is an inhibitor of tyrosine kinases and also a dual inhibitor of PDGFRβ(IC50s = 5.0 μM) and VEGFR-2 (Flk-1/KDR)(IC50s = 9.3 μM).
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产品描述Tyrphostin AG1433 is an inhibitor of tyrosine kinases and also a dual inhibitor of PDGFRβ(IC50s = 5.0 μM) and VEGFR-2 (Flk-1/KDR)(IC50s = 9.3 μM).(In Vitro):In glioblastoma cells, administration of Tyrphostin AG1433 (0.1-100 μM; 72 hours; GB8B cells) induces moderate cytotoxicity .(In Vivo):Tyrphostin AG1433 is prepared in methylcellulose pellets and applies to the CAMs of 4-6-day-old chicken embryos, and prevents the formation of new vessels under the pellets .
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同义词SU1433; AG1433
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通路Angiogenesis
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靶点VEGFR
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受体——
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研究领域——
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适应症——
化学信息
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CAS Number168835-90-3
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分子量266.3
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分子式C16H14N2O2
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纯度>98% (HPLC)
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溶解度——
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SMILESOC1=CC=C(C2=NC3=CC(C)=C(C)C=C3N=C2)C=C1O
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1.Shuyun Shi, et al. A high-speed counter-current chromatography- HPLC-DAD method for preparative isolation and purification of two polymethoxylated flavones from Taraxacum mongolicum. J Chromatogr Sc . May-Jun 2009;47(5):349-53.
产品手册
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